Andrea Rosario Beccari
Andrea Rosario Beccari
Drug Discovery Platform Manager, Dompe
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ELR+ CXC chemokines and their receptors (CXC chemokine receptor 1 and CXC chemokine receptor 2) as new therapeutic targets
C Bizzarri, AR Beccari, R Bertini, MR Cavicchia, S Giorgini, M Allegretti
Pharmacology & therapeutics 112 (1), 139-149, 2006
Targeting C5a: recent advances in drug discovery
M Allegretti, A Moriconi, AR Beccari, RD Bitondo, C Bizzarri, R Bertini, ...
Current medicinal chemistry 12 (2), 217-236, 2005
Design of noncompetitive interleukin-8 inhibitors acting on CXCR1 and CXCR2
A Moriconi, MC Cesta, MN Cervellera, A Aramini, S Coniglio, S Colagioia, ...
Journal of medicinal chemistry 50 (17), 3984-4002, 2007
Combining molecular modeling with experimental methodologies: mechanism of membrane permeation and accumulation of ofloxacin
M Fresta, S Guccione, AR Beccari, PM Furneri, G Puglisi
Bioorganic & medicinal chemistry 10 (12), 3871-3889, 2002
Receptor binding mode and pharmacological characterization of a potent and selective dual CXCR1/CXCR2 non‐competitive allosteric inhibitor
R Bertini, LS Barcelos, AR Beccari, B Cavalieri, A Moriconi, C Bizzarri, ...
British journal of pharmacology 165 (2), 436-454, 2012
Targeting the minor pocket of C5aR for the rational design of an oral allosteric inhibitor for inflammatory and neuropathic pain relief
A Moriconi, TM Cunha, GR Souza, AH Lopes, FQ Cunha, VL Carneiro, ...
Proceedings of the National Academy of Sciences 111 (47), 16937-16942, 2014
LiGen: a high performance workflow for chemistry driven de novo design
AR Beccari, C Cavazzoni, C Beato, G Costantino
Journal of chemical information and modeling 53 (6), 1518-1527, 2013
The ANTAREX approach to autotuning and adaptivity for energy efficient HPC systems
C Silvano, G Agosta, S Cherubin, D Gadioli, G Palermo, A Bartolini, ...
Proceedings of the ACM International Conference on Computing Frontiers, 288-293, 2016
Biological and biophysical properties of the histone deacetylase inhibitor suberoylanilide hydroxamic acid are affected by the presence of short alkyl groups on the phenyl ring
F Oger, A Lecorgne, E Sala, V Nardese, F Demay, S Chevance, ...
Journal of medicinal chemistry 53 (5), 1937-1950, 2010
Molecular mechanism and functional role of brefeldin A-mediated ADP-ribosylation of CtBP1/BARS
A Colanzi, G Grimaldi, G Catara, C Valente, C Cericola, P Liberali, ...
Proceedings of the National Academy of Sciences 110 (24), 9794-9799, 2013
Allosteric inhibitors of chemoattractant receptors: opportunities and pitfalls
M Allegretti, R Bertini, C Bizzarri, A Beccari, A Mantovani, M Locati
Trends in pharmacological sciences 29 (6), 280-286, 2008
PARP1-produced poly-ADP-ribose causes the PARP12 translocation to stress granules and impairment of Golgi complex functions
G Catara, G Grimaldi, L Schembri, D Spano, G Turacchio, ML Monte, ...
Scientific reports 7 (1), 1-17, 2017
Use of experimental design to optimize docking performance: The case of ligendock, the docking module of ligen, a new de novo design program
C Beato, AR Beccari, C Cavazzoni, S Lorenzi, G Costantino
Journal of chemical information and modeling 53 (6), 1503-1517, 2013
The ANTAREX tool flow for monitoring and autotuning energy efficient HPC systems
C Silvano, G Agosta, J Barbosa, A Bartolini, AR Beccari, L Benini, J Bispo, ...
2017 International Conference on Embedded Computer Systems: Architectures …, 2017
AutoTuning and Adaptivity appRoach for Energy efficient eXascale HPC systems: the ANTAREX Approach
C Silvano, G Agosta, A Bartolini, AR Beccari, L Benini, J Bispo, R Cmar, ...
2016 Design, Automation & Test in Europe Conference & Exhibition (DATE), 708-713, 2016
Exploring the activation mechanism of TRPM8 channel by targeted MD simulations
A Pedretti, A Labozzetta, ML Monte, AR Beccari, A Moriconi, G Vistoli
Biochemical and biophysical research communications 414 (1), 14-19, 2011
Auto-regulation of secretory flux by sensing and responding to the folded cargo protein load in the endoplasmic reticulum
A Subramanian, A Capalbo, NR Iyengar, R Rizzo, A di Campli, ...
Cell 176 (6), 1461-1476. e23, 2019
(R)-arylalkylamino derivatives and pharmaceutical compositions containing them
M Allegretti, A Moriconi, A Aramini, MC Cesta, A Beccari, R Bertini
US Patent 8,026,367, 2011
Do-it-yourself lamp structure
US Patent 6,758,577, 2004
Novel selective, potent naphthyl TRPM8 antagonists identified through a combined ligand-and structure-based virtual screening approach
AR Beccari, M Gemei, ML Monte, N Menegatti, M Fanton, A Pedretti, ...
Scientific reports 7 (1), 1-15, 2017
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